Rilmenidine hemifumarate

SKU: orb2653204

Description

Rilmenidine hemifumarate, an innovative antihypertensive agent, is an orally active, selective I1 imidazoline receptor agonist. Rilmenidine hemifumarate is an alpha 2-adrenoceptor agonist. Rilmenidine hemifumarate induces autophagy. Rilmenidine hemifumarate acts both centrally by reducing sympathetic overactivity and in the kidney by inhibiting the Na+/H+ antiport. Rilmenidine hemifumarate modulates proliferation and stimulates the proapoptotic protein Bax thus inducing the perturbation of the mitochondrial pathway and apoptosis in human leukemic K562 cells .

Key Properties

• CAS Number: 207572-68-7
• MW: 476.565846443176
• Purity: >98%
• Formula: C₂₄H₃₆N₄O₆
• SMILES: C1CC1C(C2CC2)NC3=NCCO3.C1CC1C(C2CC2)NC3=NCCO3.C(=C\C(=O)O)/C(=O)O

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only