Rhapontigenin 3'-O-glucoside

SKU: orb1221594

Description

Rhapontigenin 3'-O-glucoside is a derivative of Rhapontigenin. Rhapontigenin is a potent inactivator of human P450 1A1 and is a good candidate for a cancer chemopreventive agent.

Images & Validation

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Key Properties

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CAS Number	94356-22-6
MW	420.4
Purity	>98% (HPLC)
Formula	C₂₁H₂₄O₉
SMILES	COC1=C(C=C(C=C1)/C=C/C2=CC(=CC(=C2)O)O)O[C@H]3[C@@H]([C@H]([C@@H]([C@H](O3)CO)O)O)O
Target	Dopamine Receptor
Solubility	In Vitro: DMSO : 100 mg/mL (237.86 mM)

Bioactivity

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In Vitro	Rhapontigenin exhibits a potent and selective inhibition of human P450 1A1 with an IC50 of 0.4 μM. Rhapontigenin shows 400-fold selectivity for P450 1A1 over P450 1A2 and 23-fold selectivity for P450 1A1 over P450 1B1.

Storage & Handling

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Storage	Storage temperature: -20°C. Stability: ≥ 2 years
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Quick Database Links

Gene Symbol

Dopamine Receptor

Protocol Information

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