PSMA-617 TFA

SKU: orb3033053

Description

PSMA-617, also know as vipivotide tetraxetan, is a ligand used to make 177Lu-PSMA-617, which is a radioactive molecule to fight cancer. PSMA617 possesses a small peptide, which was designed to target prostate-specific membrane antigen (PSMA). PSMA617 demonstrates high radiolytic stability for at least 72 h. PSMA617 has high inhibition potency (equilibrium dissociation constant Ki=2.34±2.94 nM on LNCaP; Ki=0.37±0.21 nM enzymatically determined). 177 Lu-PSMA-617 offers a potential additional life-prolonging treatment option for men with mCRPC.

Research Area

Immunology & Inflammation

Key Properties

• MW: 1498.25
• Purity: 0.98
• Formula: C₅₇H₇₅F₁₂N₉O₂₄

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only