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Protein kinase G inhibitor-1

SKU: orb1685590

Description

Protein kinase G inhibitor-1 is a potent and selective cGMP-dependent protein kinase (PKG) antagonist with an IC50 of 0.9 µM. It is a valuable research tool for investigating PKG signaling pathways in cardiovascular physiology, smooth muscle function, and nociception in both cellular and animal models.

Research Area

Infectious Disease & Virology, Pharmacology & Drug Discovery, Signal Transduction

Images & Validation

Key Properties

CAS Number354544-70-0
MW278.37
Purity98.64% (May vary between batches)
FormulaC14H18N2O2S
SMILESC(N)(=O)C=1C2=C(SC1NC(=O)C3CC3)CC(C)CC2
TargetPKA,Antibacterial
SolubilityDMSO:30 mg/mL (107.77 mM)

Bioactivity

Target IC50
PKG:0.9 uM

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

Protein kinase G inhibitor-1, PKG, WAY312157

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Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Protocol Information

Available Sizes

Select a size below

1 mg
$ 90.00
1 ml x 10 mM (in DMSO)
$ 150.00
5 mg
$ 160.00
10 mg
$ 210.00
25 mg
$ 290.00
50 mg
$ 390.00
100 mg
$ 510.00
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