PROTAC PIN1 degrader-1

SKU: orb2665587

Description

PROTAC PIN1 degrader-1 is a potent and selective degrader of the PIN1 protein, demonstrating a DC50 of 18 nM in MDA-MB-468 triple-negative breast cancer cells. This research compound is a valuable chemical tool for studying PIN1's role in oncology, supporting both in vitro and in vivo cancer research applications.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 3038591-59-9
• MW: 917.02
• Formula: C₅₁H₅₂N₁₀O₇
• SMILES: N#CC=1C=CC(=CC1)C2=CC=C(C=C2)N3N=NC(=C3)CC(NC(=O)C4(C5=NC=CC=C5C)CC4)C(=O)NC6CCN(CCCCCOC7=CC=CC=8C(=O)N(C(=O)C78)C9C(=O)NC(=O)CC9)CC6
• Target: PROTACs

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

172638560