PKI(5-24)

SKU: orb1679393

Description

This small molecule is a potent and selective inhibitor of protein kinase A (PKA), exhibiting a high binding affinity with a Ki of 2.3 nM. It is a valuable research tool for studying cAMP/PKA signaling pathways in both cellular (in vitro) and animal (in vivo) models of physiology and disease.

Research Area

Signal Transduction

Key Properties

• Target: PKA
• CAS Number: 99534-03-9
• MW: 1925.057
• Formula: C₇₆H₁₂₉N₃₁O₂₈
• SMILES: CCCC(NC(=O)CNC(=O)CNC(=O)CNC(=O)CNC(=O)C(NC(=O)CC(C)O)C(C)O)C(=O)NC(C)C(=O)NC(CO)C(=O)NCC(=O)NC(CCCNC(N)=N)C(=O)NC(C(C)O)C(=O)NCC(=O)NC(CCCNC(N)=N)C(=O)NC(CCCNC(N)=N)C(=O)NC(CC(N)=O)C(=O)NC(C)C(=O)NC(C(C)CC)C(=O)NC(Cc1cnc[nH]1)C(=O)NC(CC(O)=O)C(O)=O

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

71434297