PKC-iota inhibitor 1

SKU: orb1298652

Description

PKC-iota inhibitor 1 is a potent and selective small molecule targeting protein kinase C-iota (PKC-ι), exhibiting an IC50 of 0.34 µM. This compound is a valuable research tool for investigating PKC-ι signaling in cancer cell proliferation and transformation, with applications in both in vitro biochemical and cellular assays.

Research Area

Epigenetics & Chromatin, Pharmacology & Drug Discovery, Signal Transduction

Key Properties

• CAS Number: 2328094-11-5
• MW: 374.44
• Purity: 98.82% (May vary between batches)
• Formula: C₂₁H₂₂N₆O
• SMILES: Nc1ncc(cc1C(=O)Nc1ccncc1)-c1cccc(c1)N1CCNCC1
• Target: PKC,AMPK
• Solubility: DMSO:125 mg/mL (333.83 mM)

Bioactivity

• Target IC50:
  PKCι:0.34 μM

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Inhibitor, inhibit, PKC, PKC iota inhibitor 1, PKC-ι, PKCiota inhibitor 1, PKC-iota inhibitor 1, Protein kinase C

Compound Identifiers

PubChem CID

138377600