PKA-IN-1

SKU: orb1691481

Description

PKA-IN-1 is a potent and selective inhibitor of the cyclic AMP-dependent protein kinase catalytic subunit (cAK), exhibiting an IC50 of 0.03 μM. This compound is a valuable research tool for investigating PKA signaling in immune system disorders and has been utilized in both cellular and biochemical studies.

Research Area

Signal Transduction

Key Properties

• CAS Number: 179985-52-5
• MW: 225.25
• Purity: 99.12% (May vary between batches)
• Formula: C₁₃H₁₁N₃O
• SMILES: CC(=O)Nc1nc(C)c(C#N)c2ccccc12
• Target: PKA
• Solubility: 10% DMSO+90% Corn Oil:2.5 mg/mL (11.1 mM);DMSO:55 mg/mL (244.17 mM)

Bioactivity

• Target IC50:
  CAK:0.03 μM (IC50)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

PKA, PKA IN 1, PKAIN1, PKA-IN-1

Compound Identifiers

PubChem CID

3691181