PIN1 inhibitor 3

SKU: orb2664914

Description

Compound A0 is a potent PIN1 inhibitor (KD = 25 nM, IC50 = 150 nM) used as a ligand for PROTAC development. It is a valuable chemical probe for studying PIN1 function in cancer research, with applications in both in vitro biochemical assays and in vivo model studies.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 3039570-04-9
• MW: 587.71
• Formula: C₃₅H₃₇N₇O₂
• SMILES: N#CC=1C=CC(=CC1)C2=CC=C(C=C2)N3N=NC(=C3)CC(NC(=O)C4(C=5C=CC=CC5C)CC4)C(=O)NC6CCN(C)CC6
• Target: Ligands for Target Protein for PROTAC

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

172638559