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PIK75

SKU: orb1222313

Description

PIK-75 Hydrochloride is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM in cell-free assays.

Images & Validation

Key Properties

CAS Number372196-67-3
MW452.3
Purity>98% (HPLC)
FormulaC16H14BrN5O4S
TargetDNA-PK| p110α| p110β| p110γ| p110δ

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Protocol Information

PIK75 (orb1222313)

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200 mg
500 mg
5 mg
$ 80.00
10 mg
$ 100.00
25 mg
$ 180.00
50 mg
$ 290.00
100 mg
$ 490.00