PF-03382792

SKU: orb1695710

Description

PF-03382792 is a selective 5-HT4 receptor agonist used as a research tool for Alzheimer's disease. It is applied in both in vitro binding assays and in vivo models to study receptor-mediated cognitive enhancement and potential neuroprotective pathways.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1400811-63-3
• MW: 433.52
• Purity: 99.64%
• Formula: C₂₃H₃₂FN₃O₄
• SMILES: C(NCC1CCN(CC2(O)CCOCC2)CC1)(=O)N3C=4C(C(C)(C)C3=O)=CC=C(F)C4
• Target: 5-HT Receptor
• Solubility: DMSO:4.34 mg/mL (10.01 mM)

Bioactivity

• Target IC50:
  5-HT4D receptor:2.7 nM (Ki)|5-HT4D receptor:0.9 nM (EC50)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

5HTReceptor, 5-HT4, 5HT Receptor, PF03382792, PF-03382792, PF 03382792

Compound Identifiers

PubChem CID

71451950