PERK-IN-3

SKU: orb1708902

Description

PERK-IN-3 is a highly potent and selective PERK inhibitor with an IC50 of 7.4 nM. This small molecule is a valuable research tool for investigating the unfolded protein response (UPR) in cellular and animal models of diseases such as cancer and neurodegeneration.

Research Area

Cell Biology, Signal Transduction

Key Properties

• CAS Number: 1337532-08-7
• MW: 406.38
• Formula: C₂₂H₁₆F₂N₄O₂
• SMILES: NC1=C2C(=COC2=NC=N1)C=3C=C4C(=CC3)N(C(CC5=C(F)C=CC(F)=C5)=O)CC4
• Target: ERK,PERK

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

66561010