Pentagastrin

SKU: orb1302741

Description

Pentagastrin (ICI-50123) is a synthetic gastrin-like peptide used in research to stimulate gastric acid secretion. It is widely applied in physiological studies, including in vitro receptor assays and in vivo models investigating gastrointestinal function and salivary protein synthesis.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 5534-95-2
• MW: 767.89
• Purity: 99.49% (May vary between batches)
• Formula: C₃₇H₄₉N₇O₉S
• SMILES: CSCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCNC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
• Target: Cholecystokinin Receptor
• Solubility: 10% DMSO+90% Corn Oil:2 mg/mL (2.6 mM);DMSO:135 mg/mL (175.81 mM)

Bioactivity

• Target IC50:
  CCKB receptor:11 nM (IC50)

Storage & Handling

• Storage: keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Cholecystokinin Receptor, Cholecystokinin, CCK Receptor, CCKB receptor, inhibit, gastric acid, gastric mucosa, ICI50123, ICI-50123, ICI 50123, Inhibitor, Pentagastrin

Compound Identifiers

PubChem CID

9853654