PDK1-IN-RS2

SKU: orb1988990

Description

PDK1-IN-RS2 is a substrate-selective inhibitor of PDK1 (Kd: 9 μM) that mimics the PIFtide docking motif, thereby blocking PDK1-mediated activation of downstream effectors like S6K1. This cell-permeable compound is a valuable research tool for studying PI3K/PDK1 signaling in cancer and metabolic diseases in cellular models.

Research Area

Signal Transduction

Key Properties

• CAS Number: 1643958-89-7
• MW: 380.89
• Formula: C₁₅H₉ClN₂O₂S₃
• SMILES: Clc1ccc2nc(NS(=O)(=O)c3cc4ccccc4s3)sc2c1
• Target: PDK

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

86290242