Queen's Award Received in 2021 ISO 9001 Certified Delivered over 1,000,000 bio-reagents to life science researchers Trusted by Life Science Communities
Cart summary

You have no items in your shopping cart.

PDHK1-IN-1

SKU: orb2944862

Description

PDHK1-IN-1 (compound 17) is a selective PDHK1 inhibitor (IC50 = 1.5 µM) that blocks phosphorylation of PDC E1α at Ser232 and Ser293, reversing PDHK1-mediated suppression of oxidative metabolism. This tool compound is used in cancer metabolism research to study the Warburg effect and has demonstrated anticancer properties in cellular assays.

Research Area

Metabolism Research

Images & Validation

Key Properties

MW404.66
FormulaC14H11BrClNO4S
TargetDehydrogenase

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Protocol Information