PD-217014 HCl

SKU: orb1699679

Description

PD-217014 is a GABA analog that acts as a potent, nanomolar-affinity ligand (Kᵢ = 18 nM) for the alpha-2-delta subunit of voltage-gated calcium channels, inhibiting gabapentin binding. It demonstrates visceral analgesic properties in vivo, making it a useful research tool for studying neuropathic pain and calcium channel function.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 444088-20-4
• MW: 197.27
• Formula: C₁₁H₁₉NO₂
• SMILES: C(C(OC)=O)[C@@]1(CN)C[C@@]2([C@](C1)(CC2)[H])[H]
• Target: Others,Calcium Channel

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

45098889