PARP7-IN-16

SKU: orb1943224

Description

PARP7-IN-16 (compound 36) is a highly potent and selective oral inhibitor of PARP-1, PARP-2, and PARP-7 with respective IC50 values in the sub-nanomolar range. Its promising activity in preclinical models supports research into its potential therapeutic applications for cancers such as breast and prostate cancer.

Research Area

Epigenetics & Chromatin, Molecular Biology, Signal Transduction

Key Properties

• CAS Number: 2435657-10-4
• MW: 488.49
• Formula: C₂₅H₂₆FN₄NaO₄
• SMILES: O=C1[N-]C(N(CC2=CC=C(C(C(N3CC(N(C(CC)CC)CC3)=O)=O)=C2)F)C4=C1C=CC=C4)=O.[Na+]
• Target: PARP

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

169450724