PARP-1-IN-1

SKU: orb1688239

Description

PARP-1-IN-1 is a potent and selective PARP-1 inhibitor with sub-nanomolar activity (IC50 = 0.96 nM). It is orally bioavailable and has shown significant in vivo efficacy in xenograft models like MDA-MB-436, making it a valuable chemical probe for studying DNA damage response and oncology research.

Research Area

Cell Biology, Epigenetics & Chromatin, Molecular Biology

Key Properties

• MW: 392.47
• Formula: C₂₃H₂₅FN₄O
• Target: PARP,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

PARP,Others