p38α MAPK/CK1δ inhibitor-1

SKU: orb2944377

Description

Compound 3 is a dual inhibitor of p38α MAPK and CK1δ, demonstrating potent activity with IC50 values of 0.185 µM and 0.089 µM, respectively. This small molecule is a valuable research tool for studying inflammation, cancer, and circadian rhythms in both cellular and animal models.

Research Area

Metabolism Research, Pharmacology & Drug Discovery, Signal Transduction, Stem Cell & Developmental Biology

Key Properties

• CAS Number: 1572047-84-7
• MW: 440.429
• Formula: C₂₄H₁₇FN₆O₂
• SMILES: O=C(O)C1=CC=CC(=C1)N2N=NC(=C2)C3=NC(C=4C=CC(F)=CC4)=C(C=5C=CN=CC5)N3C
• Target: p38 MAPK,Casein Kinase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

76332540