P300-IN-4

SKU: orb2802538

Description

P300-IN-4 (compound 6) is a small molecule inhibitor of the histone acetyltransferase p300, exhibiting an IC50 of 12.2 µM. It serves as a research tool for probing p300's role in epigenetic regulation, cancer biology, and cellular processes in both in vitro and in vivo experimental models.

Research Area

Epigenetics & Chromatin, Metabolism Research, Signal Transduction

Key Properties

• MW: 674.91
• Formula: C₂₉H₂₈ClIN₄O₅
• SMILES: O=C1N(CC(CC2=CC=C(Cl)C=C2)C(O)=O)NC3=C1C=CC(C(N[C@H](CC(NC)=O)CC4=CC=C(I)C=C4)=O)=C3
• Target: Histone Acetyltransferase,HSP

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

176419322