P2X7 receptor antagonist-3

SKU: orb1745069

Description

P2X7 receptor antagonist-3 is a highly potent and selective small molecule inhibitor of the P2X7 receptor, with IC50 values of 4.2 nM (human) and 6.8 nM (rat). It is a valuable research tool for studying P2X7-mediated signaling in neuroinflammation, pain, and immune responses in both cellular and animal models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1627900-92-8
• MW: 408.77
• Formula: C₁₇H₁₂ClF₃N₆O
• SMILES: C(=O)(N1CC2=C(N(N=N2)C=3N=CC=CN3)CC1)C4=C(Cl)C(C(F)(F)F)=CC=C4
• Target: P2X Receptor,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

86270913