Opiranserin hydrochloride

• Catalog Number: orb1297854
• Category: Small Molecules
• Description: Opiranserin hydrochloride
• CAS Number: 1440796-75-7
• Purity: 98%
• MW: 430.97
• SMILES: Cl.CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCOCC1)N(C)C
• Formula: C₂₁H₃₅ClN₂O₅
• Biological Activity: Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 μM). It is development as an injectable agent for the treatment of postoperative pain.
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.