OMDM-5

SKU: orb1309299

Description

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU, Ki=4.8 µM) and a potent TRPV1 agonist (EC50=75 nM), with weak affinity for the CB1 receptor (Ki=4.9 µM). This pharmacological profile makes it a useful research tool for studying endocannabinoid and vanilloid signaling pathways in vitro.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 616884-66-3
• MW: 432.64
• Purity: 99.72%
• Formula: C₂₆H₄₄N₂O₃
• SMILES: C(NNC(CCCCCCC/C=C\CCCCCCCC)=O)C1=CC(OC)=C(O)C=C1
• Target: Endogenous Metabolite,Cannabinoid Receptor,TRP/TRPV Channel
• Solubility: DMSO:65 mg/mL (150.24 mM)

Bioactivity

• Target IC50:
  CB1:4.9 μM(Ki)|ACU:4.8 μM(Ki)|TRPV1:75 Nm(TRPV1)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

cannabinoid, Cannabinoid Receptor, CannabinoidReceptor, anandamide cellular uptake, acids, cells, CB2, CB1, Endogenous Metabolite, EndogenousMetabolite, fatty, FAAH, Inhibitor, Human Endogenous Metabolite, inhibit, OMDM 5, OMDM5, OMDM-5, RBL-2H3, receptor, type, vanilloid, uptake, TRP Channel, Transient receptor potential channels, TRPVChannel, TRPV Channel, TRPV1, TRPChannel, VR1

Compound Identifiers

PubChem CID

146026184