Olcegepant hydrochloride

SKU: orb1708988

Description

Olcegepant hydrochloride is a potent and selective antagonist of the CGRP1 receptor, exhibiting an IC50 of 0.03 nM and a Ki of 14.4 pM. It is widely used in research to investigate CGRP-mediated pathways in migraine pathophysiology, utilizing both in vitro binding assays and in vivo animal models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 586368-06-1
• MW: 906.11
• Formula: C₃₈H₄₈Br₂ClN₉O₅
• SMILES: Cl.NCCCC[C@H](NC(=O)[C@@H](Cc1cc(Br)c(O)c(Br)c1)NC(=O)N1CCC(CC1)N1Cc2ccccc2NC1=O)C(=O)N1CCN(CC1)c1ccncc1
• Target: Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

9919272