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MZ82

SKU: orb2695576

Description

MZ82 is a potent and brain-penetrant ABCG2/BCRP inhibitor (IC50 ~23 nM), derived from Ko 143. It demonstrates superior metabolic stability in liver microsomes and improved in vivo performance in mice, making it a valuable tool for studying drug efflux and pharmacokinetics in cancer and neuroscience research.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

MW431.53
FormulaC26H29N3O3
TargetBCRP

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

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Protocol Information

MZ82 (orb2695576)

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Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

Step 2: Enter the in vivo formulation

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