MRS542

SKU: orb1739138

Description

MRS542 acts as an A3 adenosine receptor (A3AR) antagonist in cAMP assays but demonstrates partial agonist activity in β-arrestin translocation assays, a property attributed to the presence of LUF6000. This unique functional selectivity makes it a valuable tool for studying biased signaling in both in vitro and in vivo models of inflammation, ischemia, and cancer.

Key Properties

• CAS Number: 163152-31-6
• MW: 517.71
• Formula: C₁₇H₁₇ClIN₅O₄
• SMILES: N(CC1=CC(I)=CC=C1)C2=C3C(N(C=N3)[C@@H]4O[C@H](CO)[C@@H](O)[C@H]4O)=NC(Cl)=N2
• Target: Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

10346511