MRGPRX4 modulator-3

SKU: orb3173216

Description

MRGPRX4 modulator-3 (Compound 1C) is an allosteric negative modulator of MAS-related G-protein coupled receptor X4 (MRGPRX4). It significantly inhibits the activation response induced by Nateglinide (an orthosteric agonist), with an IC50 of 337 nM. MRGPRX4 modulator-3 is applicable in studies related to chronic itching, particularly cholestatic pruritus, and pain.

Images & Validation

−

Key Properties

−

Target	MRGPR

Storage & Handling

−

Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Quick Database Links

Gene Symbol

MRGPR

Documents Download

Datasheet

Product Information

Download

Request a Document

Protocol Information

Find More Protocols