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ML-109

SKU: orb1309411

Description

ML-109

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1186649-91-1
MW523.58
Purity98.14% (May vary between batches)
FormulaC31H29N3O5
SMILESCOc1ccc(cc1COc1ccc(NC(C)=O)cc1)C1Nc2cccc(O)c2C(=O)N1Cc1ccccc1
TargetTSH Receptor
SolubilityDMSO:83.33 mg/mL (159.15 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (6.3 mM)

Bioactivity

Target IC50
TSHR:40 nM(EC50)
In Vitro
ML-109 is a full agonist at TSHR with an EC50 of 40 nM ,has no activity at FSHR or LHCGR.

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

thyrotropin receptor (TSHR), Thyrotropin receptor, Thyroid-stimulating hormone Receptor, TSH Receptor, TSHReceptor, inhibit, ML 109, ML109, ML-109, Inhibitor

Similar Products

  • ML-109 [orb1220122]

    >98% (HPLC)

    1186649-91-1

    523.58

    C31H29N3O5

    5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 2 mg, 200 mg, 500 mg, 1 g
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Key Properties

No computed properties available.

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Protocol Information

ML-109 (orb1309411)

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

1 mg
$ 80.00
2 mg
$ 90.00
5 mg
$ 120.00
1 ml x 10 mM (in DMSO)
$ 130.00
10 mg
$ 170.00
25 mg
$ 290.00
50 mg
$ 440.00
100 mg
$ 640.00
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