MEK1 Derived Peptide Inhibitor 1

SKU: orb1980887

Description

This cell-permeable peptide inhibitor selectively blocks MEK1-mediated activation of ERK2 with an IC50 of 30 µM. It is a valuable tool for investigating MAPK/ERK signaling pathways in both in vitro biochemical assays and cellular research models.

Research Area

Pharmacology & Drug Discovery, Signal Transduction

Key Properties

• Target: ERK,MEK
• CAS Number: 355367-87-2
• MW: 1491.84
• Formula: C₆₈H₁₁₈N₁₈O₁₇S
• SMILES: CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N1CCC[C@H]1C(O)=O

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

10214285