MCH(human, mouse, rat) TFA

SKU: orb1981608

Description

MCH (human, mouse, rat) TFA is a potent peptide agonist for MCH receptors, exhibiting binding IC50 values of 0.3 nM for MCH1R and 1.5 nM for MCH2R. It is particularly effective against MCH-2R in a CHO cell line, with functional activation EC50 values of 3.9 nM for MCH-1R and 0.1 nM for MCH-2R, as evidenced by intracellular calcium mobilization measured with FLIPR.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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MW	2500.86
Formula	C₁₀₇H₁₆₁F₃N₃₀O₂₈S₄
Target	Melanin-concentrating Hormone Receptor (MCHR),GPCR

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Gene Symbol

Melanin-concentrating Hormone Receptor (MCHR),GPCR

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