Cart summary

You have no items in your shopping cart.

mAChR antagonist 1

SKU: orb1942878

Description

Compound 4a is a muscarinic acetylcholine receptor (mAChR) antagonist with subtype selectivity, exhibiting Ki values of 121 nM (M3), 158 nM (M4), 255 nM (M1), and 255 nM (M5). This tool compound is suitable for in vitro binding assays and functional studies to investigate cholinergic signaling pathways in neurological and metabolic research.

Research Area

Neuroscience

Images & Validation

Key Properties

CAS Number101491-79-6
MW310.39
FormulaC19H22N2O2
SMILESO=C(OC1CCN(C)CC1)N(C=2C=CC=CC2)C=3C=CC=CC3
TargetOthers,AChR

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Similar Products

  • mAChR-IN-1 hydrochloride [orb1301614]

    99.83%

    119391-73-0

    524.82

    C23H26ClIN2O2

    5 mg, 10 mg, 1 mg, 25 mg, 50 mg, 100 mg, 200 mg, 1 ml x 10 mM (in DMSO)
  • Pirenzepine dihydrochloride [orb1308257]

    99.68%

    29868-97-1

    424.32

    C19H21N5O2·2HCl

    1 ml x 10 mM (in H2O), 1 g, 500 mg, 100 mg
  • Anisodine [orb1740330]

    99.28%

    52646-92-1

    319.35

    C17H21NO5

    50 mg, 25 mg, 1 mg, 5 mg, 10 mg
  • Solifenacin [orb1299178]

    99.91% (May vary between batches)

    242478-37-1

    362.46

    C23H26N2O2

    25 mg, 50 mg, 100 mg, 500 mg, 1 ml x 10 mM (in DMSO)
  • mAChr-in-1 [orb1689881]

    119391-56-9

    488.36

    C23H25IN2O2

    1 ml x 10 mM (in DMSO), 25 mg
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Documents Download

Datasheet
Product Information
Download

Request a Document

Protocol Information

mAChR antagonist 1 (orb1942878)

  • Star
  • Star
  • Star
  • Star
  • Star
  • 0.0
Based on 0 reviews

Participating in our Biorbyt product reviews program enables you to support fellow scientists by sharing your firsthand experience with our products.

Login to Submit a Review

No reviews yet

Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

Step 2: Enter the in vivo formulation

(This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO +
%+
% Tween 80 +
%