LPAR1 antagonist 2

SKU: orb2565864

Description

LPAR1 antagonist 2 (example 76) is a potent small molecule inhibitor of the lysophosphatidic acid receptor 1, demonstrating an average IC50 of 130 nM. This antagonist is a valuable research tool for studying LPA1-mediated pathways in fibrosis, cancer, and pain in both cellular and animal models.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1664336-46-2
• MW: 409.86
• Formula: C₂₃H₂₀ClNO₄
• SMILES: C(N(CC1=CC=C(C(O)=O)C=C1)CC)(=O)C2=CC=C(OC3=C(Cl)C=CC=C3)C=C2
• Target: LPL Receptor,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

117903669