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LEI-101

SKU: orb1700164

Description

LEI-101 is a potent and selective oral cannabinoid CB2 receptor agonist, exhibiting high affinity for human CB2 (pEC50 8) with minimal hERG inhibition. Its ~100-fold CB2/CB1 selectivity supports research into inflammatory and oxidative stress-related pathologies, such as kidney disease, in both in vitro and in vivo experimental models.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1228660-00-1
MW472.53
FormulaC23H25FN4O4S
SMILESO=C1N(C(=O)CN1CC2=CC=C(C=C2)C=3N=C(CN4CCS(=O)(=O)CC4)C(F)=CC3)C5CC5
TargetOthers,Cannabinoid Receptor

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

LEI-101 (orb1700164)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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