Laniquidar

SKU: orb1685907

Description

Laniquidar (R101933) is a potent third-generation, non-competitive P-glycoprotein inhibitor with an IC50 of 0.51 µM. It is utilized in research to study and overcome multidrug resistance in cancer cell models, though its in vivo application is limited by poor oral bioavailability.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 197509-46-9
• MW: 584.71
• Formula: C₃₇H₃₆N₄O₃
• SMILES: C(OC)(=O)C=1N2C(C(C=3C(CC2)=CC=CC3)=C4CCN(CCC5=CC=C(OCC6=NC7=C(C=C6)C=CC=C7)C=C5)CC4)=NC1
• Target: Others,P-gp

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

6450806