KSK94 FA

SKU: orb1980150

Description

KSK94 FA is a selective and potent histamine H3 receptor antagonist used in research. It is employed in both in vitro binding assays and in vivo models to investigate its potential roles in neuropathic pain and obesity-related studies.

Research Area

Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• MW: 444.53
• Purity: 98.68% (May vary between batches)
• Formula: C₂₆H₂₈N₄O₃
• SMILES: N#CC1=CC=C(C2=CC=C(C=C2)OCCCN3CCN(CC3)C4=CC=NC=C4)C=C1.[H]C(O)=O
• Target: Histamine Receptor

Bioactivity

• Target IC50:
  H3 receptor:7.9 nM|Sigma 2 Receptor:75.2 nM|Sigma 1 Receptor:2958 nM

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

KSK94 FA(2566716-07-0 Free base), KSK94FA(2566716070Freebase), H3 receptor, Histamine Receptor, HistamineReceptor

Compound Identifiers

PubChem CID

171361083