KSK68

SKU: orb1944241

Description

KSK68 is a potent dual sigma-1 receptor and histamine H3 receptor antagonist with high affinity, exhibiting potential analgesic activity. It is a valuable research tool for investigating pain mechanisms in both in vitro and in vivo experimental models.

Research Area

Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2566715-91-9
• MW: 364.48
• Purity: 99.11% (May vary between batches)
• Formula: C₂₃H₂₈N₂O₂
• SMILES: O=C(C1=CC=C(OCCCN2CCC(C=3C=CN=CC3)CC2)C=C1)C4CC4
• Target: Histamine Receptor,Sigma receptor

Bioactivity

• Target IC50:
  σ1 receptor:3.6 nM|H3 receptor:7.7 nM|σ2 receptor:22.4 nM

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

H3 receptor, Histamine Receptor, HistamineReceptor

Compound Identifiers

PubChem CID

162643335