Keap1-Nrf2-IN-3

SKU: orb1691253

Description

Keap1-Nrf2-IN-3 is a potent small molecule inhibitor that disrupts the KEAP1-NRF2 protein-protein interaction, exhibiting high affinity with a Kd of 2.5 nM for KEAP1. This compound is a valuable research tool for studying the NRF2 pathway in oxidative stress and inflammation models, applicable in both cellular and animal studies.

Research Area

Cancer Biology, Immunology & Inflammation

Key Properties

• CAS Number: 2095066-47-8
• MW: 538.652
• Formula: C₃₁H₃₄N₆O₃
• SMILES: CCC[C@@H]1CCCCN1C(=O)c1cccc(c1)-c1cccc(c1)-n1ncc(C(O)=O)c1[C@@H]1C[C@H]1c1cn(C)nn1
• Target: Nrf2,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

126754534