KDM4-IN-2

SKU: orb1709344

Description

KDM4-IN-2 is a potent, dual inhibitor of KDM4 and KDM5 histone demethylases, exhibiting high selectivity with Kis of 4 nM for KDM4A and 7 nM for KDM5B. This small molecule is a valuable chemical probe for epigenetic research, enabling the study of histone methylation roles in cancer and other diseases in cellular and biochemical assays.

Research Area

Epigenetics & Chromatin, Metabolism Research

Key Properties

• CAS Number: 2369607-62-3
• MW: 426.51
• Formula: C₂₅H₂₆N₆O
• SMILES: O=c1[nH]cnc2c(nccc12)-n1cc(CCN2CCC3(CCc4ccccc34)CC2)cn1
• Target: Histone Demethylase,Glucokinase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

138393336