KDM1/CDK1-IN-1

SKU: orb1687639

Description

KDM1/CDK1-IN-1 is a dual inhibitor of KDM1 and CDK1 with sub-micromolar potency. It induces G2/M cell cycle arrest and apoptosis, demonstrating cytotoxic effects in various cancer cell lines such as CCRF-CEM, HOP-92, and Hep-G2. This compound is a useful chemical probe for oncology research, particularly in studying cell cycle regulation and epigenetic modulation in vitro.

Research Area

Cell Biology, Epigenetics & Chromatin, Metabolism Research; Cell Biology, Protein Biochemistry

Key Properties

• MW: 431.47
• Formula: C₂₂H₁₇N₅O₃S
• Target: Histone Demethylase,Others,CDK,Apoptosis,Caspase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Histone Demethylase,Others,CDK,Apoptosis,Caspase