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JNJ-63533054

SKU: orb1223228

Description

JNJ 63533054 is a potent and selective GPR139 agonist (EC50 = 16 nM) that is brain and cell penetrant. JNJ 63533054 is selective for GPR139 over a panel of GPCRs, ion channels and transporters, including GPR142 and is orally bioavailable.

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Key Properties

CAS Number1802326-66-4
MW316.78
Purity>98% (HPLC)
FormulaC17H17ClN2O2
SMILESC[C@@H](c1ccccc1)NC(=O)CNC(=O)c1cc(ccc1)Cl
TargetAdrenergic Receptor
SolubilityDMSO : ≥ 50 mg/mL 157.84 mM; H2O : < 0.1 mg/mL

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

JNJ 63533054 | JNJ63533054 | JNJ-63533054

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  • JNJ-63533054 [orb1304517]

    >99.99% (May vary between batches)

    1802326-66-4

    316.78

    C17H17ClN2O2

    10 mg, 25 mg, 50 mg, 100 mg, 1 mg, 5 mg, 200 mg, 1 ml x 10 mM (in DMSO)
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JNJ-63533054 (orb1223228)

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Available Sizes

Select a size below

5 mg
$ 110.00
10 mg
$ 150.00
25 mg
$ 280.00
50 mg
$ 470.00
100 mg
$ 690.00
500 mg
$ 1,410.00