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Catalog Number | orb1709508 |
---|---|
Category | Small Molecules |
Description | GYKI 52466 dihydrochloride |
CAS Number | 2319722-40-0 |
Purity | 98.00% |
MW | 366.24 |
SMILES | CC1=NN=C(C2=CC=C(N)C=C2)C3=C(C=C4OCOC4=C3)C1.Cl.Cl |
Formula | C17H17Cl2N3O2 |
Biological Activity | GYKI 52466 dihydrochloride is orally active and non-competitive kainate- and AMPA-activated currents antagonist (IC50s: 7.5 μM and 11 μM). It is inactive against NMDA or γ-aminobutyric acid responses. It is a muscle relaxant and anticonvulsant agent and has good blood-brain barrier permeability. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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