GXH-II-052

SKU: orb1982514

Description

GXH-II-052 is a potent bivalent BET inhibitor with high affinity for BRD4 and BRDT domains, exhibiting sub-nanomolar to low nanomolar Kd values. It demonstrates antiproliferative activity and suppresses c-Myc expression in vitro, making it a valuable chemical probe for oncology and epigenetics research.

Research Area

Epigenetics & Chromatin

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Key Properties

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MW	1366.39
Formula	C₆₂H₇₆Cl₂F₂N₁₄O₁₁S₂
Target	Epigenetic Reader Domain,Others

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Gene Symbol

Epigenetic Reader Domain,Others

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GXH-II-052

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