GSK2807 Trifluoroacetate

SKU: orb1219293

Description

GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM).GSK2807, a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). A high-resolution crystal structure reveals that GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3.

Key Properties

• CAS Number: 2245255-66-5
• MW: 566.5
• Purity: >98% (HPLC)
• Formula: C₂₁H₃₃F₃N₈O₇
• Target: SMYD3

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

SMYD3