GSK256066

• Catalog Number: orb1301115
• Category: Small Molecules
• Description: GSK256066
• CAS Number: 801312-28-7
• Purity: 99.66%
• MW: 518.58
• SMILES: N(C=1C2=C(C(C)=CC(S(=O)(=O)C3=CC(C(N(C)C)=O)=CC=C3)=C2)N=CC1C(N)=O)C4=CC(OC)=CC=C4
• Formula: C₂₇H₂₆N₄O₅S
• Biological Activity: GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, > 380, 000-fold selectivity versus PDE1/2/3/5/6 and > 2500-fold selectivity against PDE4B versus PDE7.Phase 2.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.