GSK248233A

SKU: orb2566156

Description

GSK248233A is a dual-targeting small molecule inhibitor with potent activity against VEGFR2 (IC50 = 2 nM) and Firefly luciferase (Fluc; IC50 = 1.03 µM). It serves as a valuable research tool for studying angiogenesis and AGC kinase signaling, while its Fluc inhibition is a critical consideration for interpreting bioluminescence reporter assays in both cellular and animal models.

Research Area

Cardiovascular Research, Signal Transduction

Key Properties

• CAS Number: 850665-21-3
• MW: 484.51
• Formula: C₂₅H₂₄N₈O₃
• SMILES: C(C)N1C=2C(N=C1C3=NON=C3N)=CN=C(OC4=CC(NC(=O)C5=CC=C(N(C)C)C=C5)=CC=C4)C2
• Target: Others,VEGFR

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

16099859