GSK-2807 free base

SKU: orb1739742

Description

GSK2807 is a potent, selective, and SAM-competitive SMYD3 inhibitor (Ki = 14 nM) that occupies both the cofactor and substrate-binding sites. It has demonstrated anti-proliferative effects in cancer cell lines and has been utilized as a chemical probe to investigate SMYD3's role in oncology and epigenetics research.

Research Area

Epigenetics & Chromatin

Key Properties

• CAS Number: 2245255-65-4
• MW: 452.51
• Formula: C₁₉H₃₂N₈O₅
• SMILES: O[C@H]1[C@H](N2C=3C(N=C2)=C(N)N=CN3)O[C@H](CN(CC[C@@H](C(O)=O)N)CCCN(C)C)[C@H]1O
• Target: Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

118797898