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GRL-03022

SKU: orb3174365

Description

GRL-03022 is a potent and highly selective non-covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), with an IC50 of 60 nM. It demonstrates over 16,000-fold selectivity for GRK5 compared to GRK2 (IC50 > 1000 μM). GRL-03022 is applicable in research related to heart failure and cancer.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

TargetGRK

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

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Protocol Information