GRK2i TFA

SKU: orb1981521

Description

GRK2i TFA is a cell-permeable inhibitory polypeptide that acts as a specific Gβγ antagonist by mimicking its binding domain, thereby blocking Gβγ-mediated GRK2 activation. This tool compound is widely used in cardiovascular and oncology research to study GPCR signaling pathways in both cellular and animal models.

Research Area

Immunology & Inflammation, Pharmacology & Drug Discovery

Key Properties

• Target: GRK
• MW: 3598.1
• Formula: C₁₅₂H₂₅₇F₃N₅₀O₄₃S

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

GRK