Grapiprant

• Catalog Number: orb1296072
• Category: Small Molecules
• Description: Grapiprant
• CAS Number: 415903-37-6
• Purity: 99.49%
• MW: 491.61
• SMILES: C(C)C=1N(C=2C(N1)=C(C)N=C(C)C2)C3=CC=C(CCNC(NS(=O)(=O)C4=CC=C(C)C=C4)=O)C=C3
• Formula: C₂₆H₂₉N₅O₃S
• Biological Activity: Grapiprant (AAT-007) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM).
• Note: For research use only
• Expiration Date: 12 months from date of receipt.