GR 89696 fumarate

SKU: orb1704507

Description

GR 89696 fumarate is a potent and selective κ2 opioid receptor agonist (IC50 = 0.04 nM). It exhibits anti-pruritic, anti-injury, and neuroprotective properties, making it a valuable research tool for studying pain, itch, and neuroprotection in both in vitro and in vivo models.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 126766-32-3
• MW: 530.4
• Purity: 99.84% (May vary between batches)
• Formula: C₂₃H₂₉Cl₂N₃O₇
• SMILES: C(=C/C(O)=O)\C(O)=O.C(CC1=CC(Cl)=C(Cl)C=C1)(=O)N2C(CN3CCCC3)CN(C(OC)=O)CC2
• Target: Opioid Receptor
• Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.77 mM);DMSO:45 mg/mL (84.84 mM);Ethanol:3.6 mg/mL (6.79 mM);H2O:7.7 mg/mL (14.52 mM)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

κ-opioid receptor, GR89696 Fumarate, GR-89696 Fumarate, GR 89696 Fumarate, GR 89696 fumarate, OpioidReceptor, Opioid Receptor

Compound Identifiers

PubChem CID

6442840